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  5. Tocris Bioscience™ Pelitinib

Tocris Bioscience™ Pelitinib

Product Code. 18759066
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25 mg
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25mg
5mg
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18759066 25 mg 25mg
18787856 5 mg 5mg
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Product Code. 18759066 Supplier Tocris Bioscience™ Supplier No. 6349/25

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Description

Potent and irreversible EGFR inhibitor (IC50 = 20-80 nM); orally bioavailable

Pelitinib is a potent irreversible EGFR inhibitor (IC50 = 20-80 nM). Selective for EGFR over Src, MEK/ERK, erbB2, Raf, c-Met and Cdk4 (IC50 values are 282, 800, 1255, 3353, 4100 and >20,000). Inhibits the growth of tumors overexpressing EGFR in vivo. Orally bioavailable.
TRUSTED_SUSTAINABILITY

Specifications

Chemical Name or Material (2E)-N-[4-[(3-Chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxy-6-quinolinyl]-4-(dimethylamino)-2-butenamide
CAS 257933-82-7
Synonym EKB-569
Quantity 25 mg
Molecular Formula C24H23ClFN5O2
Formula Weight 467.92
Purity 97%
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