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GSK2801, MedChemExpress

Product Code. 16462807
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16462807 50 mg 50mg
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Product Code. 16462807 Supplier Medchem Express Supplier No. HY15658

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Description

MedChemExpress GSK2801 is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4.

GSK2801 is a potent, selective, orally active and cell active acetyl-lysine competitive BAZ2A and BAZ2B bromodomains inhibitor with Kd values of 136 nM and 257 nM, respectively. GSK2801 shows >50-fold selectivity for BAZ2A/B over BRD4.

Specifications

Chemical Name or Material GSK2801
CAS 1619994-68-1
Color Light Yellow
Purity Grade Notes Research
Molecular Formula C20H21NO4S
Quantity 50 mg
Solubility Information DMSO : 50 mg/mL (134.61 mM; Need ultrasonic)
SMILES O=C(C)C1=CC(C2=C(S(=O)(C)=O)C=CC=C2)=C3N1C=CC(OCCC)=C3
Molecular Weight (g/mol) 371.45
Formula Weight 371.45
Percent Purity 95.0%
Grade Research
Physical Form Solid
For Use With (Application) Cancer-programmed cell death
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Research purposes only

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