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Brexpiprazole, MedChemExpress

Product Code. 16471786
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Product Code. 16471786 Supplier Medchem Express Supplier No. HY15780

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Description

MedChemExpress Brexpiprazole (OPC-34712), an atypical orally active antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).

Brexpiprazole (OPC-34712), an atypical orally active antipsychotic drug, is a partial agonist of human 5-HT1A and dopamine D2L receptor with Kis of 0.12 nM and 0.3 nM, respectively. Brexpiprazole is also a 5-HT2A receptor antagonist with a Ki of 0.47 nM. Brexpiprazole also shows potent antagonist activity at human noradrenergic α1B (Ki=0.17 nM) and α2C receptors (Ki=0.59 nM).

Specifications

Chemical Name or Material Brexpiprazole
CAS 913611-97-9
Color White
Purity Grade Notes Research
Molecular Formula C25H27N3O2S
Quantity 500 mg
Synonym OPC-34712
Solubility Information DMSO : 25 mg/mL (57.66 mM; ultrasonic and warming and heat to 80°C)
SMILES O=C1NC2=C(C=CC(OCCCCN3CCN(C4=C(C=CS5)C5=CC=C4)CC3)=C2)C=C1
Molecular Weight (g/mol) 433.57
Formula Weight 433.57
Percent Purity 98.25%
Grade Research
Physical Form Powder
For Use With (Application) Neuroscience-Neuromodulation
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Research purposes only

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