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Zamicastat, MedChemExpress

Product Code. 16466767
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Product Code. 16466767 Supplier Medchem Express Supplier No. HY106004

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Description

MedChemExpress Zamicastat (BIA 5-1058) is a dopamine β-hydroxylase (DBH) inhibitor and can cross the blood-brain barrier (BBB) to cause central as well as peripheral effects. Zamicastat is also a concentration-dependent dual P-gp and BCRP inhibitor with IC50 values of 73.8 μM and 17.0 μM, respectively. Zamicastat reduces high blood pressure.

Zamicastat (BIA 5-1058) is a dopamine β-hydroxylase (DBH) inhibitor and can cross the blood-brain barrier (BBB) to cause central as well as peripheral effects. Zamicastat is also a concentration-dependent dual P-gp and BCRP inhibitor with IC50 values of 73.8 μM and 17.0 μM, respectively. Zamicastat reduces high blood pressure.

Specifications

Chemical Name or Material Zamicastat
CAS 1080028-80-3
Color Off-White
Purity Grade Notes Research
Molecular Formula C21H21F2N3OS
Quantity 5 mg
Synonym BIA 5-1058
Solubility Information DMSO : 150 mg/mL (373.63 mM; Need ultrasonic)
SMILES S=C1N([C@@H]2CC3=CC(F)=CC(F)=C3OC2)C(CCNCC4=CC=CC=C4)=CN1
Molecular Weight (g/mol) 401.47
Formula Weight 401.47
Percent Purity 95.36%
Grade Research
Physical Form Solid
For Use With (Application) Cancer-programmed cell death
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Research purposes only

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