CAS RN 37025-55-1
CAS RN 37025-55-1
Carbetocin, TRC
CAS: 37025-55-1 Synonym: Glycinamide, N-(4-mercapto-1-oxobutyl)-O-methyl-L-tyrosyl-L-isoleucyl-L-glutaminyl-L-asparaginyl-L-cysteinyl-L-prolyl-L-leucyl-, cyclic (1→5)-thioether∣1-Carbaoxytocin, 1-butanoic acid-2-(O-methyl-L-tyrosine)- (9CI)∣1-Thia-4,7,10,13,16-pentaazacycloeicosane, cyclic peptide deriv.∣Carbetocin∣Deamino-2-O-methyltyrosine-1-carbaoxytocin∣Depotocin∣Duratocin∣Pabal∣[2-O-Methyltyrosine]-deamino-1-carba-oxytocin∣[Desamino-monocarba1,Tyr(methyl)2]-oxytocin
Carbetocin, MedChemExpress
MedChemExpress Carbetocin, an oxytocin (OT) analogue, is an oxytocin receptor agonist with a Ki of 7.1 nM. Carbetocin has high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 μM). Carbetocin has the potential for postpartum hemorrhage research. Carbetocin can crosse the blood-brain barrier and produces antidepressant-like activity via activation of oxytocin receptors in the CNS.